Found 48 of ec50 data for polymerid = 10494 
Affinity DataEC50: 6.30nMAssay Description:Agonist activity at MF1 mouse brain CB1 receptor assessed as induction of [35S]GTPgammaS binding after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 7.5nMT: 2°CAssay Description:[35S]GTPγS binding was performed as previously described [Brents et al., PLoS One, 6:e21917]. Briefly, 25 μg of mouse brain homogenates were...More data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Activity at CB1 receptor assessed as stimulation of [35S]GTP-gamma-S binding in DBA/J2 mouse brainMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Activity at CB1R in mouse brain membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding preincubated for 60 mins prior to [35S]GT...More data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Positive allosteric modulation of CB1 receptor in MF1 mouse vas deferens assessed as inhibition of AEA-induced electrically evoked vas deferens contr...More data for this Ligand-Target Pair
Affinity DataEC50: 42nMAssay Description:Agonist activity at MF1 mouse brain CB1 receptor assessed as induction of [35S]GTPgammaS binding after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataEC50: 77nMT: 2°CAssay Description:[35S]GTPγS binding was performed as previously described [Brents et al., PLoS One, 6:e21917]. Briefly, 25 μg of mouse brain homogenates were...More data for this Ligand-Target Pair
Affinity DataEC50: 78.4nMAssay Description:Agonist activity at MF1 mouse brain CB1 receptor assessed as induction of [35S]GTPgammaS binding after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 113nMT: 2°CAssay Description:[35S]GTPγS binding was performed as previously described [Brents et al., PLoS One, 6:e21917]. Briefly, 25 μg of mouse brain homogenates were...More data for this Ligand-Target Pair
Affinity DataEC50: 138nMAssay Description:Activity at CB1 receptor assessed as stimulation of [35S]GTP-gamma-S binding in DBA/J2 mouse brainMore data for this Ligand-Target Pair
Affinity DataEC50: 204nMAssay Description:Activity at CB1 receptor assessed as stimulation of [35S]GTP-gamma-S binding in DBA/J2 mouse brainMore data for this Ligand-Target Pair
Affinity DataEC50: 277nMT: 2°CAssay Description:[35S]GTPγS binding was performed as previously described [Brents et al., PLoS One, 6:e21917]. Briefly, 25 μg of mouse brain homogenates were...More data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Agonist activity at CB1 receptor in mouse brain membrane assessed as stimulation of GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 820nMAssay Description:Agonist activity at CB1 receptor in Swiss Webster mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 940nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.45E+3nMAssay Description:Agonist activity at CB1 receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+3nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.73E+3nMAssay Description:Agonist activity at CB1 receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataEC50: >6.00E+3nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.44E+3nMAssay Description:Agonist activity at CB1 receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 8.99E+3nMAssay Description:Agonist activity at CB1 receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse CB1 receptor by cAMP read-out assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.19E+4nMAssay Description:Agonist activity at CB1 receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 1.35E+4nMAssay Description:Agonist activity at CB1 receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at mouse recombinant CB1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
Affinity DataEC50: 3.69E+4nMAssay Description:Agonist activity at CB1 receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 3.69E+4nMAssay Description:Agonist activity at CB1 receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 3.84E+4nMAssay Description:Agonist activity at CB1 receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
